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Sugammadex Sodium

An injection that reverses muscle relaxation from rocuronium or vecuronium after surgery.

Clinical information

Common uses

  • reversing rocuronium or vecuronium muscle relaxation after surgery

Common side effects

  • vomiting
  • pain
  • feeling sick
  • low blood pressure
  • headache

Cautions

  • serious allergic reactions (anaphylaxis) can occur
  • marked slow heart rate, rarely cardiac arrest
  • not recommended with severe kidney impairment

Interactions

  • toremifene — can delay recovery
  • hormonal contraceptives — use extra non-hormonal contraception for 7 days

Pregnancy: limited data — no clear risk identified

Reference information, not medical advice — always follow your doctor or pharmacist. Source: DailyMed, dailymed.nlm.nih.gov, sugammadex sodium label, setid 0379799d-b678-4eb1-8f15-7dd183ee2a6e (accessed 2026-08-16)

Approved brands & formulations1

Brand nameDosage formStrengthImporterCategory
Sugammadex SodiumParenteral ( Injection- Solution )100mg/mlMFDA designated importers with Pre Authorization approval before importhospital
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