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Sitagliptin + Metformin

A combination tablet of sitagliptin and metformin that lowers blood sugar in type 2 diabetes.

Clinical information

Common uses

  • type 2 diabetes, alongside diet and exercise

Common side effects

  • diarrhoea
  • upper respiratory tract infection
  • headache

Cautions

  • boxed warning: lactic acidosis risk, especially with kidney problems
  • pancreatitis can occur — stop if suspected
  • may lower vitamin B12 levels
  • not for type 1 diabetes

Interactions

  • carbonic anhydrase inhibitors, e.g. topiramate, acetazolamide
  • drugs that reduce metformin clearance, e.g. cimetidine, dolutegravir
  • alcohol — raises lactic acidosis risk
  • insulin or insulin secretagogues — low blood sugar risk

Pregnancy: only if prescribed — talk to your doctor

Reference information, not medical advice — always follow your doctor or pharmacist. Source: DailyMed, dailymed.nlm.nih.gov, Zituvimet (sitagliptin and metformin) label, setid 0098dec4-f0e5-45d5-8aa4-5d0faf9ab142 (accessed 2026-08-16)

Approved brands & formulations7

Brand nameDosage formStrengthImporterCategory
Glipita-M 50/500Tablet ( Film coated )50MG+ 500MGauthorized importers after registration of the productPOM
Sitagliptin Phosphate +Metformin HclTablet50mg + 1000mgPOM
Sitagliptin Phosphate+Metformin HclTablet50mg+500mgPOM
Sita - MetTablet ( Film coated )50 mg+ 500 mg (BP)State Trading Organization PlcPOM
Swizglipt MTablet ( Film coated )50 mg (USP) + 500 mg (USP)AMDC Pvt. LtdPOM
Swizglipt M forteTablet ( Film coated )50mg (USP) + 1000mg (USP)AMDC Pvt. LtdPOM
Taglimet 50/500Tablet ( Film coated )50MG+ 500MGauthorized importers after registration of the productPOM
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