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Nilotinib

Nilotinib is a targeted cancer tablet for Philadelphia chromosome-positive chronic myeloid leukaemia.

Clinical information

Common uses

  • chronic myeloid leukaemia (Ph+ CML)

Common side effects

  • feeling sick
  • rash
  • headache
  • tiredness
  • itching

Cautions

  • boxed warning: dangerous heart rhythm changes; sudden deaths reported
  • not for people with low potassium/magnesium or long QT syndrome
  • regular ECGs and blood monitoring needed
  • can harm an unborn baby — use effective contraception

Interactions

  • strong CYP3A inhibitors — avoid or reduce dose
  • strong CYP3A inducers — avoid
  • other QT-prolonging medicines — avoid

Pregnancy: can harm an unborn baby — avoid

Reference information, not medical advice — always follow your doctor or pharmacist. Source: DailyMed, dailymed.nlm.nih.gov, nilotinib (Cavhanza) label, setid 98b197ea-bca4-427e-8737-97f70a3262bc (accessed 2026-08-16)

Approved brands & formulations2

Brand nameDosage formStrengthImporterCategory
TasignaCapsule200 mgMediquip Maldives Pvt. LtdPOM
TasignaCapsule150 mgMediquip Maldives Pvt. LtdPOM
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