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Esmolol

Fast-acting beta blocker infusion for short-term control of rapid heart rate.

Clinical information

Common uses

  • fast heart rhythms (atrial fibrillation, atrial flutter, sinus tachycardia)
  • fast heart rate and high blood pressure around surgery

Common side effects

  • low blood pressure
  • sweating
  • dizziness

Cautions

  • can cause low blood pressure, slow heart rate or heart failure
  • may worsen asthma or reactive airway disease
  • can mask low blood sugar symptoms in diabetes
  • not with severe slow heart rate, heart block or cardiogenic shock

Interactions

  • IV verapamil-type calcium blockers (fatal cardiac arrests reported)
  • digoxin (slow heart rate risk)
  • clonidine-type blood pressure drugs (rebound hypertension on stopping)
  • adrenaline-type stimulant drugs (avoid)
  • succinylcholine or mivacurium (prolonged muscle blockade)

Pregnancy: only if the benefit justifies the risk

Reference information, not medical advice — always follow your doctor or pharmacist. Source: DailyMed, dailymed.nlm.nih.gov, esmolol hydrochloride injection label, setid 01ad7942-99c3-40ee-9cfb-272fb6c44e2b (accessed 2026-08-16)

Approved brands & formulations1

Brand nameDosage formStrengthImporterCategory
EsmololParenteral ( Injection )10mg/mlMFDA designated importers with Pre Authorization approval before importhospital
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